Jahresbibliographie 2000

Veröffentlichungen von
Angehörigen der Hochschulen des Saarlandes

Pharmazeutische und Medizinische Chemie (07.06.01)

Hartmann, Rolf W.
- 1-Imidazolyl(alkyl) substituted di- and tetrahydroquinolines and analogs.
Synthesis and evaluation of dual inhibitors of P450 TxA2 and P450arom / von C.
Jacobs; Martin Frotscher; G. Dannhardt; Rolf W. Hartmann. - In: J. Med. Chem,
43 (2000), S. 1841-1851
 
- 5alpha-reductase in intact DU145 cells: Evidence for isozyme I and
evaluation of novel inhibitors / von Wolfgang Reichert; Joachim Jose; Rolf W.
Hartmann. - In: Arch. Pharm. Pharm. Med. Chem, 333 (2000), S. 201-204
 
- 6-Substituted 1H-quinolin-2-ones and 2-methoxy-quinolines: Synthesis and
evaluation as inhibitors of steroid 5alpha-reductases type 1 and 2 / von E.
Baston; A. Palusczak; Rolf W. Hartmann. - In: Eur. J. Med. Chem, 35 (2000), S.
931-940
 
- Development of a simple and rapid test assay for inhibitors of human 17a-
hydroxylase-C17,20-lyase by coexpression of cytochrome P450c17 and NADPH-
cytochrome-P450 reductase in Escherichia coli / von Peter Bernhard Ehmer;
Joachim Jose; Rolf W. Hartmann. - In: Journal of Steroid Biochemistry and
Molecular Biology, 75 (2000), 1, S. 57-63
 
- Development of a simple and rapid assay for the evaluation of inhibitors
of human 17alpha-hydroxylase-C17,20-lyase (P450c17) by coexpression of P450c17
with NADPH-cytochrome-P450-reductase in Escherichia coli / von P.B. Ehmer;
Joachim Jose; Rolf W. Hartmann. - In: J. Steroid Biochem. Mol. Biol, 75
(2000), S. 57-63
 
- Development of an improved in vitro model to study the adhesion of tumor
cells to the basement membrane / von Alice Kleber; Rolf W. Hartmann; Joachim
Jose. - In: Pharm. Pharmcol. Lett, 10 (2000), 2, S. 55-58
 
- New nonsteroidal steroid 5alpha-reductase inhibitors. Syntheses and
structure-activity-studies on carboxamide phenylalkyl-substituted pyridones
and piperidones / von Rolf W. Hartmann; Martin Reichert. - In: Arch. Pharm.
Pharm. Med. Chem, 333 (2000), S. 145-153
 
- Novel imidazolyl and triazolyl substituted biphenyl compounds: Synthesis
and evaluation as nonsteroidal inhibitors of human 17a-hydroxylase-C17,20-
lyase(P450 17) / von Y. Zhuang; B.G. Wachall; Rolf W. Hartmann. - In: Bioorg.
Med. Chem, 8 (2000), S. 1245-1252
 
- Synthesis and biological evaluation of indole derivatives acting as anti-
inflammatory or antitumoral drugs / von M. Le Brogne; M. Duflos; G. Le Baut;
P.J. Nicholls; Rolf W. Hartmann. - In: Ann. Pharm. Fr, 58 (2000), S. 316-320
 
- Synthesis and evaluation of novel steroidal oximes as inhibitors of P450
17 (17alpha-hydroxylase / C17-20-lyase) and . - a-reductase 1 and 2 / von Rolf
W. Hartmann; Markus Hector; S. Haidar; P. Ehmer; Joachim Jose. - In: J. Med.
Chem, 43 (2000), S. 4266-4277
 
- Synthesis and evaluation of 17-aliphatic heterocycle substituted steroidal
inhibitors of 17alpha-hydroxylase/C17-20-lyase(P450 17) / von Rolf W.
Hartmann; Markus Hector; B.G. Wachall; A. Palusczak; M. Palzer; Volker Huch;
Michael Veith. - In: J. Med. Chem, 43 (2000), S. 4437-4445
 
- Synthesis of N-substitued piperidine-4-(benzylidene-4-carboxylic acids)
and evaluation as inhibitors of steroid-5 alpha-reductase type 1 and 2 / von
F. Picard; E. Baston; Wolfgang Reichert; Rolf W. Hartmann. - In: Bioorg. Med.
Chem, 8 (2000), S. 1479-1487
 
Jose, Joachim
- 5alpha-reductase in intact DU145 cells: Evidence for isozyme I and
evaluation of novel inhibitors / von Wolfgang Reichert; Joachim Jose; Rolf W.
Hartmann. - In: Arch. Pharm. Pharm. Med. Chem, 333 (2000), S. 201-204
 
- Development of a simple and rapid test assay for inhibitors of human 17a-
hydroxylase-C17,20-lyase by coexpression of cytochrome P450c17 and NADPH-
cytochrome-P450 reductase in Escherichia coli / von Peter Bernhard Ehmer;
Joachim Jose; Rolf W. Hartmann. - In: Journal of Steroid Biochemistry and
Molecular Biology, 75 (2000), 1, S. 57-63
 
- Development of a simple and rapid assay for the evaluation of inhibitors
of human 17alpha-hydroxylase-C17,20-lyase (P450c17) by coexpression of P450c17
with NADPH-cytochrome-P450-reductase in Escherichia coli / von P.B. Ehmer;
Joachim Jose; Rolf W. Hartmann. - In: J. Steroid Biochem. Mol. Biol, 75
(2000), S. 57-63
 
- Development of an improved in vitro model to study the adhesion of tumor
cells to the basement membrane / von Alice Kleber; Rolf W. Hartmann; Joachim
Jose. - In: Pharm. Pharmcol. Lett, 10 (2000), 2, S. 55-58
 
- Human T cell response to meningococcal IgA 1 protease associated alpha-
proteins / von Joachim Jose; Uwe Wölk; Dirk Lorenzen; Holger Wenschuh; Thomas
F. Meyer. - In: Scandinavian Journal of Immunology, 51 (2000), S. 176-184
 
- Synthesis and evaluation of novel steroidal oximes as inhibitors of P450
17 (17alpha-hydroxylase / C17-20-lyase) and . - a-reductase 1 and 2 / von Rolf
W. Hartmann; Markus Hector; S. Haidar; P. Ehmer; Joachim Jose. - In: J. Med.
Chem, 43 (2000), S. 4266-4277
 
Kallmayer, Hans-Jörg
- 2-Amino-5,6-dihydro-1,4-benzochinon-Derivate / von Hans-Jörg Kallmayer;
Martin Doerr. - In: Scientia Pharmaceutica, 68 (2000), S. 87-100
 
- 4-Alkylamino-1,2-anthrachinone / von Hans-Jörg Kallmayer; Udo Bock. - In:
Pharmazie, 54 (1999), S. 467-468
 
- 4-Methoxy-5,6,7,8-tetrahydro-1,2-naphthochinon-1-arylhydrazone / von Hans-
Jörg Kallmayer; Udo Bock. - In: Pharmazie, 54 (1999), S. 355-358
 
- Kondensation des 4-Di-n-propylamino-1,2-anthrachinons mit Arylhydrazinen
in Methanol/Schwefelsaeure / von Hans-Jörg Kallmayer; Udo Bock. - In:
Pharmazie, 53 (1998), S. 418-420
 
- Die Umsetzung von Furosemid, Quimethazin und Hydrochlorothiazid mit Thymol
und Natriumhypochlorit / von Hans-Jörg Kallmayer; Roger Bender. - In:
Pharmazie, 55 (2000), S. 320-321
 
Kleber, Alice
- Development of an improved in vitro model to study the adhesion of tumor
cells to the basement membrane / von Alice Kleber; Rolf W. Hartmann; Joachim
Jose. - In: Pharm. Pharmcol. Lett, 10 (2000), 2, S. 55-58
 
Reichert, Wolfgang
- 5alpha-reductase in intact DU145 cells: Evidence for isozyme I and
evaluation of novel inhibitors / von Wolfgang Reichert; Joachim Jose; Rolf W.
Hartmann. - In: Arch. Pharm. Pharm. Med. Chem, 333 (2000), S. 201-204
 
- Synthesis of N-substitued piperidine-4-(benzylidene-4-carboxylic acids)
and evaluation as inhibitors of steroid-5 alpha-reductase type 1 and 2 / von
F. Picard; E. Baston; Wolfgang Reichert; Rolf W. Hartmann. - In: Bioorg. Med.
Chem, 8 (2000), S. 1479-1487